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I |
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V |
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VII |
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IX |
1. Einführung
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1 |
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6 |
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14 |
2. Rezeptortheorien — Beschreibung von Alternativen oder von Teilaspekten eines komplexen Mechanismus?
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21 |
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26 |
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29 |
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34 |
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35 |
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36 |
3. Methoden zur Charakterisierung von Membranrezeptoren durch Messung der Ligandwirkung auf isolierte Organe
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39 |
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40 |
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41 |
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41 |
4. Stereoselektivität der Interaktion von Membranrezeptoren mit Liganden
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43 |
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44 |
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47 |
5. Wie können Rezeptoren im Gewebe und in der Zelle lokalisiert werden?
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50 |
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52 |
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53 |
6. Die experimentellen Verfahren zur Charakterisierung von Membranrezeptoren durch Radioligand-Bindungsstudien
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55 |
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63 |
7. Quantitative Analyse der Ligand-Bindungskinetik
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81 |
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82 |
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88 |
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91 |
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96 |
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96 |
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97 |
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100 |
8. Die Zellmembran als Mikromilieu von Rezeptoren
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104 |
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109 |
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112 |
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114 |
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116 |
9. Aufklärung der molekularen Struktur von Rezeptoren
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125 |
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133 |
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139 |
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144 |
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148 |
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151 |
10. Rekonstitution von isolierten Membranrezeptoren in Lipidmembranen
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159 |
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168 |
11. Die Grundprinzipien der Signalweiterleitung
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175 |
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175 |
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179 |
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180 |
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180 |
12. Kopplungsglieder zwischen Rezeptoren und Effektorsystemen: Die GTP-bindenden Proteine
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185 |
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185 |
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187 |
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187 |
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189 |
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190 |
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191 |
13. Die intrazelluläre Signalweiterleitung
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193 |
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206 |
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213 |
14. Die extrazelluläre chemische Signalweiterleitung: Der Arachidonsäuremetabolismus
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222 |
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222 |
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224 |
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228 |
15. Die intrazelluläre elektrochemische Signalweiterleitung: Die Ionenkanäle der Zellmembran
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230 |
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231 |
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232 |
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236 |
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242 |
16. Funktionsstörungen von Membranrezeptoren als Krankheitsursache
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244 |
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249 |
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250 |
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252 |
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278 |